N -benzoyl- and N -sulfonyl-1,5-benzodiazepines: Comparison of their atropisomeric and conformational properties

DOI: 10.1021/jo5008509

Source and publish data:

Journal of Organic Chemistry p. 5717 - 5727 (2014)

Update date:2022-08-05

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Authors:

Yoneda, Tetsuya

Tabata, Hidetsugu

Nakagomi, Jun

Tasaka, Tomohiko

Oshitari, Tetsuta

Takahashi, Hideyo

Natsugari, Hideaki

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Article abstract of DOI:10.1021/jo5008509

The atropisomeric and conformational properties of 1,5-benzodiazepines with an N-sulfonyl (p-tosyl/mesyl) group (IIa/b) were investigated by comparison with those of the N-benzoyl congeners (I). Similar to I, when the Ar-N(SO ₂) axis was frozen

Full text of DOI:10.1021/jo5008509

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