Journal of Medicinal Chemistry p. 1340 - 1354 (2018)
Update date:2022-08-03
Topics: Inhibitors Derivatives Potent Selective Reversible 1,5-Diphenylpyrazole-3-Carboxamide Monoacylglycerol Lipase (MAGL)
Aghazadeh Tabrizi, Mojgan
Baraldi, Pier Giovanni
Baraldi, Stefania
Ruggiero, Emanuela
De Stefano, Lucia
Rizzolio, Flavio
Di Cesare Mannelli, Lorenzo
Ghelardini, Carla
Chicca, Andrea
Lapillo, Margherita
Gertsch, Jürg
Manera, Clementina
Macchia, Marco
Martinelli, Adriano
Granchi, Carlotta
Minutolo, Filippo
Tuccinardi, Tiziano
Monoacylglycerol lipase (MAGL) is a serine hydrolase that plays an important role in the degradation of the endocannabinoid neurotransmitter 2-arachidonoylglycerol, which is implicated in many physiological processes. Beyond the possible utilization of MA
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