Bioorganic and Medicinal Chemistry Letters p. 451 - 456 (1996)
Update date:2022-07-30
Topics:
Kerrigan, John E.
Shirley, Jennifer J.
Derivatives of 2-[(alkylsulfonyl)oxy]-1H-isoindole-1,3(2H)-diones (N-sulfonyloxy)phthalimides) with ring substituents in the 6-position were found to exhibit enhanced inhibitory potency and selectivity for HLE. The most potent inhibitor of HLE in this ser
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