Bioorganic and Medicinal Chemistry Letters p. 1241 - 1246 (1996)
Update date:2022-08-03
Topics:
Baraldi, Pier Giovanni
Beria, Italo
Cacciari, Barbara
Cozzi, Paolo
Franzetti, Cristina
Mongelli, Nicola
Romagnoli, Romeo
Spalluto, Giampiero
Several distamycin derivatives were synthesized from deformyl distamycin by coupling with different azole carboxylic acids bearing an alkylating moiety. Some of them showed good activities in vitro and in vivo against L 1210 murine leukemia.
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