Benzothiazepine CGP37157 and its 2′-isopropyl analogue modulate Ca2+ entry through CALHM1

DOI: 10.1016/j.neuropharm.2015.02.016

Source and publish data:

Neuropharmacology p. 503 - 510 (2015)

Update date:2022-08-05

Topics:

Authors:

Moreno-Ortega, Ana J.

Martínez-Sanz, Francisco J.

Lajarín-Cuesta, Rocío

De Los Rios, Cristóbal

Cano-Abad, María F.

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Article abstract of DOI:10.1016/j.neuropharm.2015.02.016

CALHM1 is a Ca²⁺ channel discovered in 2008, which plays a key role in the neuronal electrical activity, among other functions. However, there are no known efficient blockers able to modulate its Ca²⁺ handling ability. We herein desc

Full text of DOI:10.1016/j.neuropharm.2015.02.016

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