New chiral non-racemic piperidine-derived epoxy lactams

DOI: 10.1016/0957-4166(96)00317-5

Source and publish data:

Tetrahedron Asymmetry p. 2501 - 2504 (1996)

Update date:2022-08-03

Topics:

Authors:

Amat, Mercedes

Llor, Nuria

Hidalgo, Jose

Bosch, Joan

Molins, Elies

Miravitlles, Carles

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Article abstract of DOI:10.1016/0957-4166(96)00317-5

The preparation of the chiral non-racemic epoxy lactams 3a and 3b from the respective oxazolopiperidones 1 and the conversion of 3b to the enantiopure piperidine-derived α,β-epoxy alcohol 6 is reported.

Full text of DOI:10.1016/0957-4166(96)00317-5

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