New chiral non-racemic piperidine-derived epoxy lactams

DOI: 10.1016/0957-4166(96)00317-5

Source and publish data:

Tetrahedron Asymmetry p. 2501 - 2504 (1996)

Update date:2022-08-03

Topics:

Authors:

Amat, Mercedes

Llor, Nuria

Hidalgo, Jose

Bosch, Joan

Molins, Elies

Miravitlles, Carles

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/0957-4166(96)00317-5

The preparation of the chiral non-racemic epoxy lactams 3a and 3b from the respective oxazolopiperidones 1 and the conversion of 3b to the enantiopure piperidine-derived α,β-epoxy alcohol 6 is reported.

Full text of DOI:10.1016/0957-4166(96)00317-5

Products guided by the article

Product name:(1aS,2aS,5R,6aS)-6-Oxo-5-phenyl-tetrahydro-1,3-dioxa-5a-aza-cyclopropa[f]indene-6a-carboxylic acid benzyl ester

Cas No:182957-44-4

R&D Labs maybe for 182957-44-4

SYN Pharma Co., Ltd

Contact:86-21 60347964

Address:No.1304, West Meilong Road, Minhang District, Shanghai, China
Shenyang Mole pharmaceutical Technology Development Co.,Ltd

Contact:+86-24-31204918/13889278616

Address:No.44, wanliutang road, shenhe District of Shenyang
SHANXI XINTIANYUAN PHARMACEUTICAL CO., LTD.

website:http://www.tychemical.com

Contact:0086-358-3521713 3521715

Address:No. 1 Yintong Road, Shanxi Jiaocheng Economic Development Zone, Xiajiaying Town, Jiaocheng County, Lvliang City, Shanxi Province, China
Changyi Xinxing Technology Development Co., Ltd.

Contact:0086-510-86651065(Time Zone:8),86651656

Address:94 Yingbinxilu WestRoad, Huangtu Town, Jiangyin City, Jiangsu, China
WUHU HUAHAI BIOLOGY ENGINEERING CO LTD

Contact:+86-553-3836920

Address:7/F NO.82 LAODONG ROAD WUHU CHINA

Relevant to this article

A versatile preparation of 2-methyleneoxetanes

Doi:10.1021/jo9611733
(1996)
Chlorobis(η⁵-methylcyclopentadienyl)-(2,3,4,5, 6-pentafluorophenyl)titanium(IV)

Doi:10.1107/S0108270196006981
()
Stereocontrolled preparation of spirocyclic ethers by intramolecular trapping of oxonium ions with allylsilanes

Doi:10.1021/jo961306k
(1996)
Doi:10.1016/S0040-4039(01)89617-9
(1967)
Late-Stage Lead Diversification Coupled with Quantitative Nuclear Magnetic Resonance Spectroscopy to Identify New Structure-Activity Relationship Vectors at Nanomole-Scale Synthesis: Application to Loratadine, a Human Histamine H₁Receptor Inverse Agonist

Doi:10.1021/acs.jmedchem.0c00483
(2020)
The asymmetric Michael-type alkylation of chiral β-enamino esters: Critical role of a benzyl ester group in the racemization of adducts

Doi:10.1016/j.tetasy.2005.10.034
(2005)

Article Doi