An enantioselective synthesis of cyclopentyl-l-aspartic acid amenable to large scale

DOI: 10.1055/s-1997-1518

Source and publish data:

Synthesis p. 32 - 34 (1997)

Update date:2022-08-03

Topics:

Authors:

Moss, Neil

Ferland, Jean-Marie

Goulet, Sylvie

Guse, Ingrid

Malenfant, Eric

Plamondon, Louis

Plante, Raymond

Déziel, Robert

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1055/s-1997-1518

A new enantioselective synthesis of cyclopentyl-L-aspartic acid [(S)α-amino-1-(carboxy)cyclopentaneacetic acid] (1) and its N-Boc derivative 2 has been developed. This synthesis is amenable to kilogram scale preparation and avoids low temperature reactions and column chromatography.

Full text of DOI:10.1055/s-1997-1518

Products guided by the article

Product name:1-[(S)-Cyano-((S)-1-phenyl-ethylamino)-methyl]-cyclopentanecarboxylic acid methyl ester

Cas No:186375-13-3

R&D Labs maybe for 186375-13-3

Hangzhou Eastbiopharm Co.,Ltd.

Contact:+86-571-88931780

Address:Hangzhou,China
Mollt Biochem Co., Ltd(expird)

Contact:+86-21-38682181

Address:shanghai ,china
WD Silicone Co., Ltd

Contact:+86-27-87204219, +86-27-87215023

Address:2402, HuiGu Space-time Building, 8 Forest Road, East Lake Hi-Tech Development Zone
AllyChem Co., Ltd., Dalian, China（BBChem）

Contact:+86-411-62313318/62313328

Address:No.5 of Jinbin Road, Jinzhou New District, Dalian City, Liaoning Province, P.R.China
Kaymossy BioChem Tech Co., Ltd

website:http://www.kaimosi.com

Contact:0571-87191913/0571-87199097

Address:Room 215, Building 3rd, No.288 Ningxia Road, Qingdao city, China

Relevant to this article

Synthesis of a pentasaccharide corresponding to the repeating unit of the exopolysaccharide from Cryptococcus neoformans serovar D

Doi:10.1016/S0968-0896(96)00164-2
(1996)
Doi:10.1080/00220480309595225
(1956)
A Thermodynamic Preference of Chiral N-Methanesulfonyl and N-Arenesulfonyl 2,3-cis-3-Alkyl-2-Vinylaziridines over Their 2,3-Trans-Isomers: Useful Palladium(0)-Catalyzed Equilibration Reactions for the Synthesis of (E)-Alkene Dipeptide Isosteres

Doi:10.1021/jo961760o
(1997)
Tetrahedral Silicon-Centered Dibenzoylmethanatoboron Difluorides: Synthesis, Crystal Structure, and Photophysical Behavior in Solution and the Solid State

Doi:10.1002/cplu.201900732
(2020)
Doi:10.1007/BF00907221
()
New potent inhibitors of trypanothione reductase from Trypanosoma cruzi in the 2-aminodiphenylsulfide series

Doi:10.1016/S0223-5234(97)84360-7
(1997)

Article Doi