Synthesis and chemical reactivity of 5-methoxy-2-vinyl-4-azaindoles

Article abstract of DOI:10.1080/00397919708006075

2-Vinyl-4-azaindoles are less reactive with dienophiles than 2-vinylindoles. 5-Methoxy-2-vinyl-4-azaindole 2a and its 1-methyl derivative 2a reacts with N-phenylmaleimide to yield cycloadducts only under vigorous conditions. 2b produces a cycloadduct with

Full text of DOI:10.1080/00397919708006075

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Synthetic Communications: An
International Journal for Rapid
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Organic Chemistry
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Synthesis and Chemical
Reactivity of 5-Methoxy-2-
vinyl-4-azaindoles
Lourdes Rodriguez-Salvador a , Elena Zaballos-Garcia
a , Eugenia Gonzalez-Rosende a , Mohamed Djebouri
Sidi a , José Sepúlveda-Arques a & R. Alan Jones b
a Departament de Quimica Organica , Facultat de
Farmàcia, Universitat de València , Av Vicent Andréa
Estellés, 46100, Burjassot, València, Spain
b School of Chemical Sciences , University of East
Anglia , Norwich, NR4 7TJ, UK
Published online: 22 Aug 2006.
To cite this article: Lourdes Rodriguez-Salvador , Elena Zaballos-Garcia , Eugenia
Gonzalez-Rosende , Mohamed Djebouri Sidi , José Sepúlveda-Arques & R. Alan Jones
(1997) Synthesis and Chemical Reactivity of 5-Methoxy-2-vinyl-4-azaindoles, Synthetic
Communications: An International Journal for Rapid Communication of Synthetic
Organic Chemistry, 27:8, 1439-1447, DOI: 10.1080/00397919708006075
To link to this article: http://dx.doi.org/10.1080/00397919708006075
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