Synthesis and opiate activity of pseudo-tetrapeptides containing chiral piperazin-2-one and piperazine derivatives

DOI: 10.1248/cpb.45.1940

Source and publish data:

Chemical and Pharmaceutical Bulletin p. 1940 - 1944 (1997)

Update date:2022-08-04

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Authors:

Yamashita, Tetsushi

Tsuru, Eiji

Banjyo, Eri

Doe, Matsumi

Shibata, Kozo

Yasuda, Masahide

Gemba, Munekazu

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Article abstract of DOI:10.1248/cpb.45.1940

Enantiomeric piperazin-2-one derivatives, N,N'-ethylene-bridged alanylphenylalanines (1a or 1b), were synthesized using (S)- or (R)-alanine and phenylalanine as starting materials, and were inserted into the second and third positions of enantiomeric pseu

Full text of DOI:10.1248/cpb.45.1940

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