Ring-opening of chiral N-(3,4-dihydro-4-oxoquinazolin-3-yl)-substituted aziridines (Q-substituted aziridines): Access to Q-free chirons

DOI: 10.1016/S0040-4039(97)10586-X

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Tetrahedron Letters p. 497 - 500 (1998)

Update date:2022-08-05

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Authors:

Atkinson, Robert S.

Ayscough, Andrew P.

Gattrell, William T.

Raynham, Tony M.

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Article abstract of DOI:10.1016/S0040-4039(97)10586-X

The presence of the quinazolin-4(3H)-one ring (Q*) in N-(Q*)-aziridines facilitates ring-opening by nucleophiles: removal of the Q* group from enantiopure ring-opened products gives useful chirons.

Full text of DOI:10.1016/S0040-4039(97)10586-X

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Article Doi

Ring-opening of chiral N-(3,4-dihydro-4-oxoquinazolin-3-yl)-substituted aziridines (Q*-substituted aziridines): Access to Q*-free chirons

DOI: 10.1016/S0040-4039(97)10586-X

Source and publish data: