Concise and versatile syntheses of N-arylalkylpiperidines as potential intermediates for 4-anilidopiperidine analgesics

DOI: 10.3987/COM-97-8056

Source and publish data:

Heterocycles p. 239 - 242 (1998)

Update date:2022-07-29

Topics:

Authors:

Suh, Young-Ger

Shin, Dong-Yun

Cho, Kyung-Ho

Ryu, Jae-Sang

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Article abstract of DOI:10.3987/COM-97-8056

N-Arylalkylpiperidones and N-arylalkylspiroepoxypiperidine as potential intermediates for 4-anilidopiperidine analgesics and their structural analogues have been efficiently synthesized from the simple arylalkylamines by two and three step sequences respectively.

Full text of DOI:10.3987/COM-97-8056

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