
Tetrahedron Letters p. 5947 - 5950 (1998)
Update date:2022-08-02
Topics:
Tommasi, Ruben A.
Macchia, William M.
Parker, David T.
We have developed a novel amidine synthesis that allows the preparation of heterocyclic amidines that were previously unknown and difficult to prepare by published methods. The route involves the lithiation of heterocycles by the action of n-BuLi followed
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