
Bioorganic and Medicinal Chemistry Letters p. 2689 - 2694 (1998)
Update date:2022-08-05
Topics:
De Laszlo, Stephen E.
Visco, Denise
Agarwal, Lily
Chang, Linda
Chin, Jayne
Croft, Gist
Forsyth, Amy
Fletcher, Daniel
Frantz, Betsy
Hacker, Candice
Hanlon, William
Harper, Coral
Kostura, Matthew
Li, Bing
Luell, Sylvie
MacCoss, Malcolm
Mantlo, Nathan
O'Neill, Edward A.
Orevillo, Chad
Pang, Margaret
Parsons, Janey
Rolando, Anna
Sahly, Yousif
Sidler, Kelley
Widmer, W. Rick
O'Keefe, Stephen J.
Investigation of furans, pyrroles and pyrazolones identified 3-pyridyl- 2,5-diaryl-pyrroles as potent, orally bioavailable inhibitors of p38 kinase. 3-(4-pyridyl-2-(4-fluoro-phenyl)-5-(4-methylsulfinylphenyl)-pyrrole (L- 167307)) reduces secondary paw swe
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Doi:10.1016/S1381-1169(98)00072-7
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