
Bioorganic and Medicinal Chemistry Letters p. 1063 - 1066 (1999)
Update date:2022-08-02
Topics:
Cocuzza, Anthony J.
Chidester, Dennis R.
Culp, Steven
Fitzgerald, Lawrence
Gilligan, Paul
The Suzuki reaction has been used to synthesize a variety of aryl- substituted heterocyclic antagonists of the CRH1 receptor. Examples with several different heterocyclic cores are potent CRH receptor ligands.
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