Bioorganic and Medicinal Chemistry Letters p. 3193 - 3198 (1998)
Update date:2022-07-30
Topics:
St-Denis, Yves
Augelli-Szafran, Corinne E.
Bachand, Benoit
Berryman, Kent A.
DiMaio, John
Doherty, Annette M.
Edmunds, Jeremy J.
Leblond, Lorraine
Levesque, Sophie
Narasimhan, Lakshmi S.
Penvose-Yi, Jan R.
Rubin, J. Ronald
Tarazi, Micheline
Winocour, Peter D.
Siddiqui, M. Arshad
Peptidomimetic inhibitors of general structure 1 have been prepared. Optimization of the binding affinities of these compounds through variation of the P3 hydrophobic residue is described. Selected substituted bicylic lactams displayed interesting pharmacological profiles both in vitro and in vivo.
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