Solid-phase synthesis of phenolic steroids: Towards combinatorial libraries of estradiol derivatives

DOI: 10.1016/S0040-4039(98)02640-9

Source and publish data:

Tetrahedron Letters p. 1277 - 1280 (1999)

Update date:2022-08-02

Topics:

Authors:

Tremblay, Martin R.

Poirier, Donald

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/S0040-4039(98)02640-9

The 16β-(azidopropyl) derivative of estradiol (7) was synthesized and coupled to aminomethyl resin via a photolabile o-nitrobenzyl linker. Condensation of the corresponding iminophosphorane with activated acids successfully gave amides. Photocleavage resu

Full text of DOI:10.1016/S0040-4039(98)02640-9

Products guided by the article

Product name:4-[(8R,9S,13S,14S,16S,17S)-16-(3-Azido-propyl)-13-methyl-17-(tetrahydro-pyran-2-yloxy)-7,8,9,11,12,13,14,15,16,17-decahydro-6H-cyclopenta[a]phenanthren-3-yloxymethyl]-3-nitro-benzoic acid

Cas No:220810-56-0

R&D Labs maybe for 220810-56-0

Chongqing Rong＆Quan Pharmaceutical Technology Co. , Ltd.

Contact:86-023-65268721

Address:No. 7, Manshanhong Village, Pingdingshan, Shapingba District, Chongqing Province, China
shanghai jinshan pharmaceutical Co.,Ltd

Contact:021-57363011，13681638167

Address:No. 7966 Tingfeng Road,Jinshan,Shanghai,China
Zhangjiagang Jianing Import & Export Co.,Ltd.

Contact:086-512-55379012 13913607595

Address:NO.1 Guotai North Road Zhangjiagang Economic Development Zone,215600,Jiangsu,China
Ningbo Hi-tech Zone Nice-Synth Chemical Industry Ltd.

Contact:+86-(574)-81110986

Address:No. 1210, Building 3, Wante Business Centre, Hi-tech Zone, Ningbo
AUSHUN PHARMACEUTICAL TECHNOLOGY CO,.LTD

Contact:+86-25-86883560 15951806178

Address:14 Dayingbi, Zhujiang Rd. East, Nanjing, Jiangsu, China.

Relevant to this article

Synthesis, conformational interconversion, and photophysics of tethered porphyrin-fullerene dyads with parachute topology

Doi:10.1002/chem.200900587
(2009)
Novel ROR1 inhibitor ARI-1 suppresses the development of non-small cell lung cancer

Doi:10.1016/j.canlet.2019.05.016
(2019)
Doi:10.1021/jf60140a027
(1965)
SILICON MODIFIED REDUCTION AND REDUCTIVE ALKYLATION - APPLICATION TO THE PHENANTHRENE SYSTEM

Doi:10.1016/S0040-4039(00)82108-5
(1988)
Highly stereoselective route toward the synthesis of β- and γ-amino alcohols from homochiral α- and β-amino acylsilanes as synthetic equivalents of α- and β-amino aldehydes

Doi:10.1021/jo961392o
(1996)
A Pd-catalyzed double coupling reaction to 4,5-disubstituted imidazole alkynes

Doi:10.1080/00397919908085793
(1999)

Article Doi