A nonpeptide oxytocin receptor antagonist radioligand highly selective for human receptors

DOI: 10.1016/S0014-2999(02)02048-4

Source and publish data:

European Journal of Pharmacology p. 19 - 28 (2002)

Update date:2022-07-30

Topics:

Authors:

Lemaire, Wei

O'Brien, Julie A.

Burno, Maryann

Chaudhary, Ashok G.

Dean, Dennis C.

Williams, Peter D.

Freidinger, Roger M.

Pettibone, Douglas J.

Williams Jr., David L.

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Article abstract of DOI:10.1016/S0014-2999(02)02048-4

A novel, potent nonpeptide oxytocin receptor antagonist (1-(1-(2-(2,2,2-trifluoroethoxy)-4-(1-methylsulfonyl-4-piperidinyloxy) phenylacetyl)-4-piperidinyl)-3,4-dihydro-2(1H)-quinolinone) has been identified that can be labeled to high specific activity wi

Full text of DOI:10.1016/S0014-2999(02)02048-4

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Product name:1-(1-(4-(N-tert-butyloxycarbonyl-4-piperidinyloxy)-2-(2,2,2-trifluoroethoxy)phenylacetyl)piperidin-4-yl)-3,4-dihydro-quinolin-2(1H)-one

Cas No:221286-31-3

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