Bioorganic and Medicinal Chemistry Letters p. 2209 - 2212 (2000)
Update date:2022-08-05
Topics:
Billard, William
Binch III, Herbert
Bratzler, Kristen
Chen, Lian-Yong
Crosby Jr., Gordon
Duffy, Ruth A.
Dugar, Sundeep
Lachowicz, Jean
McQuade, Robert
Pushpavanam, Pradeep
Ruperto, Vilma B.
Taylor, Lisa A.
Clader, John W.
Piperidine analogues of our previously described piperazine muscarinic antagonists are described. Piperidine analogues show a distinct structure-activity relationship (SAR) that differs from comparable piperazines. Compounds with high selectivity and impr
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