Bioorganic and Medicinal Chemistry Letters p. 29 - 32 (2004)
Update date:2022-09-26
Topics:
Ochiai, Hiroshi
Ishida, Akiharu
Ohtani, Tazumi
Kusumi, Kensuke
Kishikawa, Katuya
Obata, Takaaki
Nakai, Hisao
Toda, Masaaki
Structural optimization of pyrazolopyridine derivative 2, which is one of the newly discovered chemical leads for PDE4 inhibitors from our in-house library, was carried out successfully. The process of discovery of new orally active PDE4 inhibitors, which
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