Synthesis of partially modified retro-inverso substance P analogues and their biological activity

DOI: 10.1021/jm00356a003

Source and publish data:

Journal of Medicinal Chemistry p. 129 - 135 (1983)

Update date:2022-08-05

Topics:

Authors:

Chorev Chorev

Rubini Rubini

Gilon Gilon

Wormser Wormser

Selinger

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Article abstract of DOI:10.1021/jm00356a003

Partial retro-inverso modification of a single peptide bond was applied to pGlu-Phe-Phe-Gly-Leu-Met-NH₂ (I), a C-terminal hexapeptide analogue of the neuropeptide substance P. Two analogues with reversed peptide bonds, between the pGlu-Phe and

Full text of DOI:10.1021/jm00356a003

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