Synthesis and biological evaluation of 6-bromo-6-substituted penicillanic acid derivatives as beta-lactamase inhibitors.

DOI: 10.1016/S0014-827X(02)01261-2

Source and publish data:

Il Farmaco p. 663 - 669 (2002)

Update date:2022-08-02

Topics:

Authors:

Bedini Bedini

Balsamini

Di Giacomo

Tontini Tontini

Citterio

Giorgi Giorgi

Di Modugno

Tarzia Tarzia

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Article abstract of DOI:10.1016/S0014-827X(02)01261-2

The synthesis of a selected set of 6-bromopenicillanic acid derivatives with an additional C6 substituent is reported. All these substances were tested as inhibitors of class A and C beta-lactamase enzymes derived from Escherichia coli (TEM-1) and E. cloa

Full text of DOI:10.1016/S0014-827X(02)01261-2

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