
Bioorganic and Medicinal Chemistry Letters p. 365 - 368 (2003)
Update date:2022-08-05
Topics:
Guerrini, Remo
Rizzi, Daniela
Zucchini, Marina
Tomatis, Roberto
Regoli, Domenico
Calo', Girolamo
Salvadori, Severo
The synthesis and pharmacological activity of novel nociceptin/orphanin FQ (N/OFQ) analogues modified in the Phe1-Gly2 peptide bond are reported. The aim of the present work was to elucidate the importance of this peptide bond for th
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