Bioorganic and Medicinal Chemistry Letters p. 1527 - 1532 (1999)
Update date:2022-08-04
Topics:
Cathers, Brian E.
Schloss, John V.
We have developed a novel strategy for the preparation of tetrahedral transition state analogs for aspartic acid and metallo-proteases based upon the sulfonimidamide functional group. Our best α-des-amino dipeptide analog binds at least 100-fold tighter than the corresponding ground state structure (i.e., amide). A previously unpublished five-membered cyclic sulfonimidamide was also synthesized.
View MoreHENAN NEW BLUE CHEMICAL CO.,LTD
website:http://www.newbluechem.com
Contact:86-371-55170693/55170694
Address:Zhengzhou International Trade New Territory,Jinshui District,Zhengzhou ,China
website:http://www.lidepharma.com
Contact:+86-25-58409506
Address:N0.2-309 2/F Chungking Express Nos.36 Nathan Road，Kowloon, HK
Hefei EnliPharma Tecnology Co.,Ltd
Contact:0086-551-66399836
Address:Qing Cheng ShuiXiang Building 805, Mengcheng North Road , ShuangFeng Economic Development Zone Anhui HeFei
Zibo Linzi Darong Fine Chemical Co., Ltd(expird)
Contact:86-532-67773200; 15689126900
Address:Qidu town,Linzi district,Zibo city,Shandong province,China
Shanghai Bojing Chemical Co., Ltd.
Contact:021-37122233
Address:6F Buildiing 11,No.388,Baifu Road,District Fengxian.Shanghai, China.
Doi:10.1016/j.bmc.2004.06.019
(2004)Doi:10.1016/j.bmcl.2005.06.028
(2005)Doi:10.1016/S0040-4039(02)00134-X
(2002)Doi:10.1246/bcsj.34.1384
(1961)Doi:10.1021/jo0201023
(2002)Doi:10.1021/om050209r
(2005)
