N-(2,4,5-trihydroxyphenethyl)normetazocine, a potential irreversible inhibitor of the narcotic receptor

DOI: 10.1021/jm00215a011

Source and publish data:

Journal of Medicinal Chemistry p. 673 - 675 (1977)

Update date:2022-07-29

Topics:

Authors:

Rice Rice

Shiotani

Creveling

Jacobson

Klee Klee

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Article abstract of DOI:10.1021/jm00215a011

The reaction of N-(2,4,5-tribenzyloxyphenyl)ethyl methanesulfonate, prepared in a seven-step sequence, with normetazocine followed by hydrogenolysis of the benzyloxy-protecting groups, gave N-(2,4,5-trihydroxyphenethyl)normetazocine. This compound was pre

Full text of DOI:10.1021/jm00215a011

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