The discovery of quinoline based single-ligand human H1and H3receptor antagonists

DOI: 10.1016/j.bmcl.2016.11.022

Source and publish data:

Bioorganic and Medicinal Chemistry Letters p. 5855 - 5859 (2016)

Update date:2022-08-05

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Authors:

Procopiou, Panayiotis A.

Ancliff, Rachael A.

Gore, Paul M.

Hancock, Ashley P.

Hodgson, Simon T.

Holmes, Duncan S.

Keeling, Steven P.

Looker, Brian E.

Parr, Nigel A.

Rowedder, James E.

Slack, Robert J.

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Article abstract of DOI:10.1016/j.bmcl.2016.11.022

A novel series of potent quinoline-based human H₁and H₃bivalent histamine receptor antagonists, suitable for intranasal administration for the potential treatment of allergic rhinitis associated nasal congestion, were identified. Com

Full text of DOI:10.1016/j.bmcl.2016.11.022

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