
Journal of Medicinal Chemistry p. 154 - 159 (1981)
Update date:2022-08-05
Press
Hofmann
Eudy
Day
Greenblatt
Safir
10-(Alkylamino)thieno[3,4-b][1,5]benzoxazepines (3) and 10-(alkylamino)thieno[3,4 b][1,5]benzothiazepines (4) were prepared by derivatization of the respective lactams (7 and 8) via phosphorus pentachloride and subsequent condensation with the appropriate
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