A New Method for Stereoselective Piperidine Annulation. Directing the 2-Azonia--Sigmatropic Rearrangement by Irreversible Hydrolysis

DOI: 10.1021/jo01313a051

Source and publish data:

Journal of Organic Chemistry p. 5229 - 5230 (1980)

Update date:2022-08-04

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Authors:

Overman, Larry E.

Yokomatsu, Tsutomu

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Article abstract of DOI:10.1021/jo01313a051

A new method for stereoselective piperidine annulation is described involving the cyclization and subsequent <3,3>-sigmatropic rearrangement of (5,5-dimethoxypentyl)-3-butenylamines.

Full text of DOI:10.1021/jo01313a051

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