
Journal of Medicinal Chemistry p. 1222 - 1225 (1984)
Update date:2022-08-05
Topics:
Rodriguez, Marc
Imbach, Jean-Louis
Martinez, Jean
A series of (2-chloroethyl)nitrosourea and nitrogen mustard amino acid derivatives have been synthesized for antitumor evaluation.Reaction of an appropriate N-protected amino acid with 2-chloroethylamine followed by removal of the N-protecting group and c
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