Journal of Medicinal Chemistry p. 5995 - 6008 (2004)
Update date:2022-08-05
Topics:
Wan, Yiqian
Wallinder, Charlotta
Plouffe, Bianca
Beaudry, Hélène
Mahalingam
Wu, Xiongyu
Johansson, Berndt
Holm, Mathias
Botoros, Milad
Karlén, Anders
Pettersson, Anders
Nyberg, Fred
F?ndriks, Lars
Gallo-Payet, Nicole
Hallberg, Anders
Alterman, Mathias
The first druglike selective angiotensin II AT2 receptor agonist (21) with a Ki value of 0.4 nM for the AT2 receptor and a Ki > 10 μM for the AT1 receptor is reported. Compound 21, with a bioavailability of 20-3
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