
Bioorganic and Medicinal Chemistry Letters p. 345 - 348 (2005)
Update date:2022-09-26
Topics:
Brinner, Kristin M.
Powles, Mary Ann
Schmatz, Dennis M.
Ellman, Jonathan A.
This paper describes potent antimalarial compounds effective against a multi-drug-resistant strain of P. falciparum (Dd2) with minimized toxicity, acceptable log D values, and stability to hepatocytic metabolism. A series of compounds with potent activity
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