
Journal of Pharmacy and Pharmacology p. 192 - 196 (1996)
Update date:2022-08-03
Topics:
Derrick, Jan
Lewis, John W.
Moynihan, Humphrey A.
Broadbear, Jillian
Woods, James H.
Cinnamoyl derivatives of β-naltrexamine (β-NTA) have been prepared and evaluated as potential irreversible opioid antagonists. In receptor binding assays, isolated tissue preparations and mouse antinociception assays the p-methylcinnamoyl derivative BU42
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