Studies on 2-Aziridinecarboxylic Acid. VI. Synthesis of β-Alkoxy-α-Amino Acids via Ring-opening Reaction of Aziridine

DOI: 10.1246/bcsj.55.3049

Source and publish data:

Bulletin of the Chemical Society of Japan p. 3049 - 3050 (1982)

Update date:2022-09-26

Topics:

Authors:

Nakajima, Kiichiro

Neya, Masahiro

Yamada, Shinichi

Okawa, Kenji

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1246/bcsj.55.3049

The reaction of aziridine derivatives having a urethane-type protecting group with several alcohols in the presence of boron trifluoride etherate afford the corresponding optically pure O-alkylserine and O-alkylthreonine derivatives via a ring-opening reaction of aziridine in good yield.

Full text of DOI:10.1246/bcsj.55.3049

Products guided by the article

Product name:(2S,3S)-3-methylaziridine-1,2-dicarboxylic acid 1-benzylester 2-methyl ester

Cas No:83824-81-1

R&D Labs maybe for 83824-81-1

Tangshan Moneide Trading Co., Ltd.

Contact:+86-315-8309571

Address:2-7-420 Jidong Building Materials Commercial Center, Tangshan, Hebei, 064000 China
Zhengzhou Institute of Chiral Pharmer Research Co., Ltd.

Contact:86-371-55219111

Address:15 Floor, 2 Building, Central China Technovalley, Zhongyuan West Road
LIDE PHARMACEUTICALS LIMITED

website:http://www.lidepharma.com

Contact:+86-25-58409506

Address:N0.2-309 2/F Chungking Express Nos.36 Nathan Road，Kowloon, HK
Chongqing Yawei Fine Chemical Co.,Ltd

Contact:0086-23-62849407

Address:Ziyou village, Nanquan town, Banan district, Chongqing China
Allicon Pharmaceuticals,Inc.

Contact:+86-519-86339586，13584329896

Address:Changzhou Scientific and Education Park

Relevant to this article

Total synthesis of (±)-3-deoxy-7,8-dihydromorphine, (±)-4-methoxy-N-methylmorphinan-6-one and 2,4-dioxygenated (±)-congeners

Doi:10.1002/hlca.19820650531
(1982)
ASYMMETRIC CONJUGATE ADDITION OF ZINCATES OR CUPRATES CONTAINING AN OPTICALLY ACTIVE AZAENOLATE OF erythro-ISOPROPYLIDENE-2-METHOXY-1,2-DIPHENYLAMINE TO 2-CYCLOALKENONES

Doi:10.1016/S0040-4039(01)91370-X
(1987)
New rare-earth metal acyl pyrazolonates: Synthesis, crystals structures, and luminescence properties

Doi:10.1134/S1070328414090024
(2014)
Doi:10.1007/BF00849431
()
CIRCULAR DICHROISM OF HYDROLYSABLE TANNINS-II DEHYDROELLAGITANNINS

Doi:10.1016/S0040-4039(00)87749-7
(1982)
STEREOSELECTIVITY IN THE TRANSFER OF THE 2-(1-DIMETHYLAMINOETHYL)PHENYL GROUP, R^*, FROM LiR^*2Cu AND Li(R^*)(2-THIENYL)Cu TO ENONES

Doi:10.1016/S0040-4039(00)87717-5
(1982)

Article Doi