
Angewandte Chemie - International Edition p. 5858 - 5862 (2018)
Update date:2022-08-03
Topics:
Zhan, Bei-Bei
Li, Ya
Xu, Jing-Wen
Nie, Xing-Liang
Fan, Jun
Jin, Liang
Shi, Bing-Feng
The site-selective functionalization of unactivated C(sp3)?H bonds remains one of the greatest challenges in organic synthesis. Herein, we report on the site-selective δ-C(sp3)?H alkylation of amino acids and peptides with maleimides
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