Asymmetric α-substituted phenethylamines. II. The enantioselective synthesis of 1-aryl-2-phenylethylamines from L- and D-amino acids by means of 1,3-asymmetric induction

DOI: 10.1248/cpb.31.31

Source and publish data:

Chemical and Pharmaceutical Bulletin p. 31 - 40 (1983)

Update date:2022-08-05

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Authors:

Suzuki Suzuki

Takahashi

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Article abstract of DOI:10.1248/cpb.31.31

Optically pure (1S, 1'S)-1-aryl-N-(1'-alkyl-2'-hydroxyethyl)-2-phenylethylamines were synthesized from L-alanine, L-leucine, and L-isoleucine via (S)-2-aminoalkanols and (E)-(S)-N-(1-alkyl-2-hydroxyethyl)arylmethylideneamines. On the other hand, the amine

Full text of DOI:10.1248/cpb.31.31

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