Protecting-group-free synthesis of a dual CCK1/CCK2 receptor antagonist

DOI: 10.1039/c0ob01004a

Source and publish data:

Organic and Biomolecular Chemistry p. 2654 - 2660 (2011)

Update date:2022-07-29

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Authors:

Liu, Jing

Deng, Xiaohu

Fitzgerald, Anne E.

Sales, Zachary S.

Venkatesan, Hariharan

Mani, Neelakandha S.

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Article abstract of DOI:10.1039/c0ob01004a

In our pursuit of an efficient, protecting-group-free synthesis of the dual CCK1/CCK2 receptor antagonist 1, we have developed chemoselective conditions for sulfonamide formation reaction in pure water and a PhNMe₂ mediated carboxamide formatio

Full text of DOI:10.1039/c0ob01004a

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