A Stereoselective Synthesis of (+/-)-Actinobolamine

DOI: 10.1039/c39900001412

Source and publish data:

Journal of the Chemical Society. Chemical communications p. 1412 - 1414 (1990)

Update date:2022-07-29

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Authors:

Holmes, Andrew B.

Kee, Alexander

Ladduwahetty, Tamara

Smith, David F.

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Article abstract of DOI:10.1039/c39900001412

A three-step sequence involving an imino ester heterocycloaddition, stereoselective epoxidation of the adduct 4 and subsequent toluene-p-sulphonic acid-promoted rearrangement afforded the 6-azabicyclo<3.2.1>octane 7 in excellent overall yield; elaboration

Full text of DOI:10.1039/c39900001412

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