New potential biologically active compounds: Design and an efficient synthesis of N-substituted 4-aryl-4,6,7,8-tetrahydroquinoline-2,5(1H,3H)-diones under microwave irradiation

DOI: 10.1016/j.bmcl.2006.03.011

Source and publish data:

Bioorganic and Medicinal Chemistry Letters p. 2925 - 2928 (2006)

Update date:2022-08-02

Topics: Characterization Biological testing Purification Protection of Functional Groups Retrosynthetic analysis Structure-Activity Relationship (SAR) Studies Product Isolation Workup Lead Optimization Selection of Starting Materials Safety and Toxicity Testing Preparation of Starting Materials

Authors:

Tu, Shujiang

Zhu, Xiaotong

Zhang, Jinpeng

Xu, Jianing

Zhang, Yan

Wang, Qian

Jia, Runhong

Jiang, Bo

Zhang, Junyong

Yao, Changsheng

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Article abstract of DOI:10.1016/j.bmcl.2006.03.011

A series of N-substituted 4-aryl-4,6,7,8-tetrahydroquinoline-2,5(1H,3H)-diones were synthesized through a rapid one-pot four-component reaction under microwave irradiation. The method has the advantages of excellent yields (82-96%) and short reaction time

Full text of DOI:10.1016/j.bmcl.2006.03.011

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