Bioorganic and Medicinal Chemistry Letters p. 2591 - 2596 (2010)
Update date:2022-08-04
Topics:
Xu, Ruo
Cole, David
Asberom, Ted
Bara, Tom
Bennett, Chad
Burnett, Duane A.
Clader, John
Domalski, Martin
Greenlee, William
Hyde, Lynn
Josien, Hubert
Li, Hongmei
McBriar, Mark
McKittrick, Brian
McPhail, Andrew T.
Pissarnitski, Dmitri
Qiang, Li
Rajagopalan, Murali
Sasikumar, Thavalakulamgar
Su, Jing
Tang, Haiqun
Wu, Wen-Lian
Zhang, Lili
Zhao, Zhiqiang
A novel series of tricyclic γ-secretase inhibitors was designed and synthesized via a conformational analysis of literature compounds. The preliminary results have shown that compounds in this new series have much improved in vitro potency and in vivo pro
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