Journal of Medicinal Chemistry p. 4716 - 4730 (2019)
Update date:2022-08-15
Topics:
Zhang, Yan
Wu, Xishan
Xue, Xiaoqian
Li, Chenchang
Wang, Junjian
Wang, Rui
Zhang, Cheng
Wang, Chao
Shi, Yudan
Zou, Lingjiao
Li, Qiu
Huang, Zenghong
Hao, Xiaojuan
Loomes, Kerry
Wu, Donghai
Chen, Hong-Wu
Xu, Jinxin
Xu, Yong
We report the design, optimization, and biological evaluation of nuclear receptor RORγinverse agonists as therapeutic agents for prostate cancer treatment. The most potent compound 27 (designated as XY101) exhibited cellular activity with an IC50 View More
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