A new synthesis of aziridine-2-carboxylates: Reaction of hexahydro- 1,3,5-triazines or N-methoxymethylanilines with alkyl diazoacetates in the presence of Lewis acid

DOI: 10.1016/S0040-4020(97)10358-1

Source and publish data:

Tetrahedron p. 851 - 858 (1998)

Update date:2022-08-05

Topics:

Authors:

Ha, Hyun-Joon

Suh, Jang-Min

Kang, Kyung-Ho

Ahn, Young-Gil

Han, Oksoo

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Article abstract of DOI:10.1016/S0040-4020(97)10358-1

Aziridine-2-carboxylates were prepared from the reaction of hexahydro- 1,3,5-triazines or N-methoxymethylanilines with alkyl diazoacetates in the presence of Lewis acid catalyst in high yield.

Full text of DOI:10.1016/S0040-4020(97)10358-1

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Product name:ethyl N-phenylaziridine-2-carboxylate

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