
Tetrahedron Letters p. 8375 - 8378 (1997)
Update date:2022-08-28
Topics:
Bhalay, Gurdip
Blaney, Paul
Palmer, Vanessa H.
Baxter, Anthony D.
A general method for the construction of tetrahydro-1,4-benzodiazepine- 2-ones on solid-support has been developed utilising a cleavage-conjugate addition protocol as the key step in the design. Using this novel, methodology the synthesis of a diverse one
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