Bioorganic and Medicinal Chemistry Letters p. 527 - 532 (2007)
Update date:2022-08-22
Topics:
Sorensen, Bryan
Winn, Martin
Rohde, Jeff
Shuai, Qi
Wang, Jiahong
Fung, Steven
Monzon, Katina
Chiou, William
Stolarik, DeAnne
Imade, Hovis
Pan, Liping
Deng, Xiaoqing
Chovan, Linda
Longenecker, Kenton
Judge, Russell
Qin, Wenying
Brune, Michael
Camp, Heidi
Frevert, Ernst U.
Jacobson, Peer
Link
Potent and selective adamantane sulfone and sulfonamide inhibitors of 11-β-HSD-1 have been discovered. Selected compounds from these series have robust pharmacokinetic profiles and strongly inhibit liver, fat, and brain HSD1 for extended periods after ora
View MoreChangsha Goomoo Chemical Technology Co.Ltd
Contact:+86-731-82197655
Address:No.649,Chezhan Rd.(N),Changsha,Hunan,China
Shanghai Bocimed Pharmaceutical Co., Ltd.
website:http://www.bocimed.com
Contact:+86-21-68861632
Address:Building 1, Lane 647, Songtao Road, Zhangjiang High-Tech Park, Shanghai
Hubei Sky Lake Chemical Co., Ltd.
Contact:+86-27-87385545
Address:Te-2, Xijiao Chemical Park, Yuekou Town, Tianmen, Hubei, China.
Hangzhou Showland Technology Co., Ltd.
Contact:86-571-88920516
Address:ROOM2118,NO.553,WENSAN ROAD,HANGZHOU,CHINA
Chongqing Changfeng Chemical Co., Ltd.
website:http://www.changfengchem.com
Contact:+86-23-67896333
Address:30th Floor, Longhu Ziduxingzuo Building A, 1st Branch,YuSong Rd., Yubei District, Chongqing, China
Doi:10.1002/cctc.201501056
(2016)Doi:10.1016/S0040-4039(99)02112-7
(2000)Doi:10.1021/j100105a019
(1993)Doi:10.1016/0022-1902(71)80179-3
(1971)Doi:10.1039/c4ra05190d
(2014)Doi:10.1021/jm00340a013
(1963)