A convenient synthesis of nitrogen-containing heterocycles bearing amino substituents from heteroaryl triflates

Article abstract of DOI:10.1055/s-1997-1041

Nitrogen-containing heterocycles bearing amino substituents were prepared by the reaction of the corresponding nitrogen-containing heteroaryl triflates with amines. The reaction affords good results with primary and secondary amines, and with aliphatic and aromatic amines. The whole triflation/amination process can also be conducted as a one-pot operation.