Bioorganic and Medicinal Chemistry Letters p. 4478 - 4481 (2017)
Update date:2022-08-29
Topics:
Hattori, Takayuki
Okitsu, Koyo
Yamazaki, Norikazu
Ohoka, Nobumichi
Shibata, Norihito
Misawa, Takashi
Kurihara, Masaaki
Demizu, Yosuke
Naito, Mikihiko
We designed and synthesized hybrid molecules for a protein knockdown method based on the recognition of a His-tag fused to a protein of interest (POI). The synthesized target protein degradation inducers contained three functional moieties: a His-tag liga
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