β-Carbolines as benzodiazepine receptor ligands. 1. Synthesis and benzodiazepine receptor interaction of esters of β-carboline-3-carboxylic acid

DOI: 10.1021/jm00358a008

Source and publish data:

Journal of Medicinal Chemistry p. 499 - 503 (1983)

Update date:2022-08-28

Topics:

Authors:

Lippke Lippke

Schunack

Wenning Wenning

Muller Muller

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Article abstract of DOI:10.1021/jm00358a008

Several esters of β-carboline-3-carboxylic acid were synthesized and tested in respect to their affinity for the benzodiazepine receptor in bovine cortex membranes. Out of these derivatives, the methyl, ethyl, and n-propyl ester were clearly the most pote

Full text of DOI:10.1021/jm00358a008

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