Bioorganic and Medicinal Chemistry Letters p. 24 - 29 (2017)
Update date:2022-08-29
Topics:
Guariento, Sara
Karawajczyk, Anna
Bull, James A.
Marchini, Gessica
Bielska, Martyna
Iwanowa, Xenia
Bruno, Olga
Fossa, Paola
Giordanetto, Fabrizio
Phosphodiesterase 4 (PDE4) inhibitors have attractive therapeutic potential in respiratory, inflammatory, metabolic and CNS disorders. The present work details the design, chemical exploration and biological profile of a novel PDE4 inhibitor chemotype. A
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