A New Method for Introducing Some Active Methylene or Methine Groups to the 3-Position of Pyrrolidine or Piperidine Skeleton, and Its Application to Preparation of a Key Intermydiate for (+/-)-Eburnamonine Synthesis

DOI: 10.1246/cl.1987.1447

Source and publish data:

Chemistry Letters p. 1447 - 1450 (1987)

Update date:2022-08-25

Topics:

Authors:

Shono, Tatsuya

Matsumura, Yoshihiro

Ogaki, Masaru

Onomura, Osamu

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Article abstract of DOI:10.1246/cl.1987.1447

A new method for introducing a bis(methoxycarbonyl)methyl or 2-oxopropyl group to the 3-position of pyrrolidine or piperidine skeleton has been exploited, and this method could be used in the synthesis of a key intermediate for the (+/-)-eburnamonine synthesis.

Full text of DOI:10.1246/cl.1987.1447

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