Synthesis of orthogonally protected thioamide dipeptides for use in solid-phase peptide synthesis

DOI: 10.1016/j.tetlet.2016.10.036

Source and publish data:

Tetrahedron Letters p. 5237 - 5239 (2016)

Update date:2022-08-11

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Authors:

Manzor, Kim

Kelleher, Fintan

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Article abstract of DOI:10.1016/j.tetlet.2016.10.036

Orthogonally protected thioamide-containing dipeptides were efficiently and cleanly prepared from the precursor dipeptides using Curphey's method (P₄S₁₀, hexamethyldisiloxane (HMDO), reflux, DCM) in 67–96% isolated yield. This was in

Full text of DOI:10.1016/j.tetlet.2016.10.036

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