117459-95-7Relevant articles and documents
ANTI-ALPHAVBETA1 INTEGRIN INHIBITORS AND METHODS OF USE
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Paragraph 0696-0697, (2016/09/26)
Provided herein, inter alia, are methods and compositions for inhibiting ανβ? integrin and for treating fibrosis.
Silver-catalyzed cyclization of N-(prop-2-yn-1-yl)pyridin-2-amines
Chioua, Mourad,Soriano, Elena,Infantes, Lourdes,Jimeno, M. Luisa,Marco-Contelles, Jose,Samadi, Abdelouahid
, p. 35 - 39 (2013/02/22)
We report herein the silver-catalyzed cycloisomerization of readily available N-(prop-2-yn-1-yl)pyridine-2-amines as a new and practical method for the synthesis of differently substituted 3-methylimidazo[1,2-a]pyridines. The isomerization reactions proce
Acetylenchemie. 9. Mitt. Anellierte Imidazole aus N-Propinylamid-Vorstufen
Reisch, Johannes,Scheer, Mathias
, p. 677 - 679 (2007/10/02)
The compound 2-(N-formyl-N-prop-2'-inyl)aminopyridine was cyclised in boiling formic acid to 3-methylimidazopyridine, with 3-methylene-2H-imidazopyridine as the intermediate.Under similar conditions the 1,3-diprop-2-inylpyrimidoquinoline-2,4-dione resulted from 1-methylimidazoquinoline-4-carbonic acid-N-2-prop-2'-inylamide and from the 1-prop-2'inylbenzonaphthyridin-2-one the 1-methylbenzoimidazonaphthyridine-4,7-dione as a new ring system, was obtained.