260558-15-4Relevant academic research and scientific papers
Practical method for preparation of 2-[18F]fluoro-4-boronophenylalanine
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Paragraph 0117-0124, (2021/04/13)
2 - Containing radioactive isotopes18 F] Fluoro -4 - boronylphenylalanine18 F [FBPA] A process for the preparation of the same. [18 F-FBPA is an efficient target compound by suggesting a precursor and reaction conditions w
METHOD FOR PRODUCING 2-FLUORO-4-BORONO-L-PHENYLALANINE, AND A DERIVATIVE OF 2-FLUORO-4-BORONO-L-PHENYLALANINE
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Paragraph 0161, (2016/10/09)
The present invention provides a method for producing 2-fluoro-4-borono-L-phenylalanine, and aderivative of 2-fluoro-4-borono-L-phenylalanine. The invention is to prepare and use a compound represented by the following formula. In the formula, R1/su
INHIBITORS OF IKK-BETA SERINE-THERONINE PROTEIN KINASE
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Page/Page column 10, (2011/04/13)
Cyclopentyl(2S,4E)-2-amino-5-{3-[4-carbamoyl-5(carbamoylamino)-2-thienyl]phenyl}pent-4-enoate; Cyclopentyl 5-{3-[4-carbamoyl-5-(carbamoylamino)-2-thienyl]phenyl}-L-norvalinate; Cyclopentyl(2S,4E)-2-amino-5-{3-[4-carbamoyl-5-(carbamoylamino)-2-thienyl]-5-m
Functionalized dibenzoborepins as components of small molecule and polymeric π-conjugated electronic materials
Caruso, Anthony,Tovar, John D.
experimental part, p. 2227 - 2239 (2011/06/11)
We present the synthesis and characterization of dibenzo[b,f]borepins (DBBs) functionalized at the para and meta position with respect to the boron center in order to understand how regiochemical issues influence photophysical and electrochemical properti
BORON-CONTAINING PI-ELECTRON MATERIALS INCORPORATING FORMALLY AROMATIC AND NEUTRAL BOREPIN RINGS
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Page/Page column 73-74, (2011/10/31)
The synthesis, functionalization and characterization of borepin-based extended pi-electron molecules is disclosed. Bulky substituents shielded the vacant boron p-orbitals thus allowing synthetic manipulation and purification under ambient lab conditions.
INHIBITORS OF IKK-β SERINE-THREONINE PROTEIN KINASE
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Page/Page column 21, (2009/12/05)
Cyclopentyl (2S,4E)-2-amino-5-{3-[4-carbamoyl-5 (carbamoylamino)-2-thienyl]phenyl}pent-4-enoate; Cyclopentyl 5-{3-[4-carbamoyl-5-(carbamoylamino)-2-thienyl]phenyl}-L-norvalinate; Cyclopentyl (2S,4E)-2-amino-5-{3-[4-carbamoyl-5-(carbamoylamino)-2-thienyl]-
ASYMMETRIC MONOANTHRACENE DERIVATIVE, MATERIAL FOR ORGANIC ELECTROLUMINESCENT DEVICE AND ORGANIC ELECTROLUMINESCENT DEVICE UTILIZING THE SAME
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Page/Page column 36, (2008/06/13)
Provided are an asymmetric monoanthracene derivative having a specific structure, a material for an organic EL device comprising the above asymmetric monoanthracene derivative and an organic EL device in which an organic thin film layer comprising a single layer or plural layers including a luminescent layer is interposed between a cathode and an anode, wherein at least one of the above organic thin film layers contains the asymmetric monoanthracene derivative described above in the form of a single component or a mixed component. Provided are an organic electroluminescent (EL) device having a high luminous efficiency and a long life, an asymmetric monoanthracene derivative which materializes the same and a material for an organic EL device.
Pyrimidines and uses thereof
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, (2008/06/13)
The invention relates to pyrimidines and uses thereof, including to inhibit lysophosphatidic acid acyltransferase β (LPAAT-β) activity and/or proliferation of cells such as tumor-cells.
Synthesis, SAR, and antitumor properties of diamino-C,N-diarylpyrimidine positional isomers: Inhibitors of lysophosphatidic acid acyltransferase-β
Gong, Baoqing,Hong, Feng,Kohm, Cory,Jenkins, Scott,Tulinsky, John,Bhatt, Rama,De Vries, Peter,Singer, Jack W.,Klein, Peter
, p. 2303 - 2308 (2007/10/03)
2,4-Diamino-N4,6-diarylpyrimidines were identified as potent, isoform specific inhibitors of lysophosphatidic acid acyltransferase-β (LPAAT-β). Active inhibitors also blocked proliferation of tumor cell lines in vitro. The effect of 2j in an in
